
Composition: Glucosamine sulfate, Lidocaine hydrochloride
Form: Concentrate for intramuscular solution preparation (ampoules A and B)
Indications: Primary and secondary osteoarthritis, osteochondrosis, spondyloarthrosis.
Contraindications: Hypersensitivity to components, heart conduction disorders, acute heart failure, epilepsy history, severe liver and kidney diseases, pregnancy, lactation, under 18 years. High risk with seafood allergy.
Dosage: IM 3 ml (ampoule A + B) 3 times/week for 4–6 weeks. Prepare solution right before injection. Oral glucosamine may be used concurrently if needed.
Side effects: Flatulence, diarrhea, constipation, urticaria, itching, burning at injection site. Possible lidocaine reactions: nausea, dizziness, tongue numbness, drowsiness, allergy, heart conduction issues.
Interactions: Compatible with NSAIDs, paracetamol, corticosteroids. Lidocaine interacts with cimetidine, beta-blockers, antiarrhythmics, TCAs, phenytoin, sedatives, and neuromuscular agents. Alcohol enhances lidocaine depression.
Warnings: Skin sensitivity test required before use. Use with caution in cardiovascular diseases, bronchial asthma, glucose intolerance. Avoid driving and operating machinery during therapy.
Age restrictions: From 18 years
Pregnancy: Contraindicated during pregnancy and breastfeeding.
Country of origin: Russia
Manufacturer: Sotex
Storage conditions: Store below 25 °C, protected from light. Keep out of children’s reach.
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Read❓ Can Sustagard be combined with oral glucosamine?
💬 Yes, injections can be combined with oral glucosamine intake.
❓ Is a prescription required?
💬 Yes, it is prescription-only due to lidocaine content and parenteral administration.